Synthesis and anti-HIV activity of 2,3-diaryl-1,3-thiazolidin-4-(thi)one derivatives

Anna Carbone; Erik De Clercq; Maria Zappalà; Christophe Pannecouque; Pietro Monforte; Anna Carbone; Alba Chimirri; Anna Maria Monforte; Angela Rao

Synthesis and anti-HIV activity of 2,3-diaryl-1,3-thiazolidin-4-(thi)one derivatives

Anna Carbone, Erik De Clercq, Maria Zappalà, Christophe Pannecouque, Pietro Monforte, Anna Carbone, Alba Chimirri, Anna Maria Monforte, Angela Rao

Scienze e Tecnologie Biologiche Chimiche e Farmaceutiche

Risultato della ricerca: Article › peer review

95 Citazioni (Scopus)

Abstract

Several 2,3-diaryl-1,3-thiazolidine-4-thione derivatives and 2,3-diaryl-1,3-thiazolidin-4-ones bearing a methyl group at C-5 position have been synthesized and tested as anti-HIV agents. The results of the in vitro tests showed that some of them proved to be effective inhibitors of HIV-1 replication.

Lingua originale	Italian
pagine (da-a)	747-751
Numero di pagine	5
Rivista	IL FARMACO
Volume	57
Stato di pubblicazione	Published - 2002

All Science Journal Classification (ASJC) codes

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title = "Synthesis and anti-HIV activity of 2,3-diaryl-1,3-thiazolidin-4-(thi)one derivatives",

abstract = "Several 2,3-diaryl-1,3-thiazolidine-4-thione derivatives and 2,3-diaryl-1,3-thiazolidin-4-ones bearing a methyl group at C-5 position have been synthesized and tested as anti-HIV agents. The results of the in vitro tests showed that some of them proved to be effective inhibitors of HIV-1 replication.",

author = "Anna Carbone and {De Clercq}, Erik and Maria Zappal{\`a} and Christophe Pannecouque and Pietro Monforte and Anna Carbone and Alba Chimirri and Monforte, {Anna Maria} and Angela Rao",

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T1 - Synthesis and anti-HIV activity of 2,3-diaryl-1,3-thiazolidin-4-(thi)one derivatives

AU - Carbone, Anna

AU - De Clercq, Erik

AU - Zappalà, Maria

AU - Pannecouque, Christophe

AU - Monforte, Pietro

AU - Carbone, Anna

AU - Chimirri, Alba

AU - Monforte, Anna Maria

AU - Rao, Angela

PY - 2002

Y1 - 2002

N2 - Several 2,3-diaryl-1,3-thiazolidine-4-thione derivatives and 2,3-diaryl-1,3-thiazolidin-4-ones bearing a methyl group at C-5 position have been synthesized and tested as anti-HIV agents. The results of the in vitro tests showed that some of them proved to be effective inhibitors of HIV-1 replication.

AB - Several 2,3-diaryl-1,3-thiazolidine-4-thione derivatives and 2,3-diaryl-1,3-thiazolidin-4-ones bearing a methyl group at C-5 position have been synthesized and tested as anti-HIV agents. The results of the in vitro tests showed that some of them proved to be effective inhibitors of HIV-1 replication.

UR - http://hdl.handle.net/10447/72444

M3 - Article

SN - 0014-827X

VL - 57

SP - 747

EP - 751

JO - Farmaco

JF - Farmaco

ER -