Identification and optimization of small molecule antagonists of vasoactive intestinal peptide receptor-1 (VIPR1)

Neelam Srivastava; Arvind Mathur; Lauren E. Kayser; Tajudheen Karatt; Kumaragurubaran K; Amrita Roy; Christopher B. Cooper; Jing Chen; Sukhen Karmakar; Anuradha Gupta; Yan Kong; Lalgudi S. Harikrishnan; David S. Nirschl; Maryellen Cvijic; George L. Trainor; Michael A. Poss; Neil T. Burford; Neelam Srivastava; Tai W. Wong

Identification and optimization of small molecule antagonists of vasoactive intestinal peptide receptor-1 (VIPR1)

Neelam Srivastava, Arvind Mathur, Lauren E. Kayser, Tajudheen Karatt, Kumaragurubaran K, Amrita Roy, Christopher B. Cooper, Jing Chen, Sukhen Karmakar, Anuradha Gupta, Yan Kong, Lalgudi S. Harikrishnan, David S. Nirschl, Maryellen Cvijic, George L. Trainor, Michael A. Poss, Neil T. Burford, Neelam Srivastava, Tai W. Wong

Risultato della ricerca: Article

7 Citazioni (Scopus)

Abstract

Identification, synthesis and structure-activity relationship of small-molecule VIPR1 antagonists encompassing two chemical series are described.

Lingua originale	English
pagine (da-a)	2287-2290
Numero di pagine	4
Rivista	BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Volume	22
Stato di pubblicazione	Published - 2012

Fingerprint

All Science Journal Classification (ASJC) codes

Biochemistry
Molecular Medicine
Molecular Biology
Pharmaceutical Science
Drug Discovery
Clinical Biochemistry
Organic Chemistry

Cita questo

Srivastava, N., Mathur, A., Kayser, L. E., Karatt, T., K, K., Roy, A., Cooper, C. B., Chen, J., Karmakar, S., Gupta, A., Kong, Y., Harikrishnan, L. S., Nirschl, D. S., Cvijic, M., Trainor, G. L., Poss, M. A., Burford, N. T., Srivastava, N., & Wong, T. W. (2012). Identification and optimization of small molecule antagonists of vasoactive intestinal peptide receptor-1 (VIPR1). BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 22, 2287-2290.

Identification and optimization of small molecule antagonists of vasoactive intestinal peptide receptor-1 (VIPR1). / Srivastava, Neelam; Mathur, Arvind; Kayser, Lauren E.; Karatt, Tajudheen; K, Kumaragurubaran; Roy, Amrita; Cooper, Christopher B.; Chen, Jing; Karmakar, Sukhen; Gupta, Anuradha; Kong, Yan; Harikrishnan, Lalgudi S.; Nirschl, David S.; Cvijic, Maryellen; Trainor, George L.; Poss, Michael A.; Burford, Neil T.; Srivastava, Neelam; Wong, Tai W.

In: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, Vol. 22, 2012, pag. 2287-2290.

Risultato della ricerca: Article

Srivastava, N, Mathur, A, Kayser, LE, Karatt, T, K, K, Roy, A, Cooper, CB, Chen, J, Karmakar, S, Gupta, A, Kong, Y, Harikrishnan, LS, Nirschl, DS, Cvijic, M, Trainor, GL, Poss, MA, Burford, NT, Srivastava, N & Wong, TW 2012, 'Identification and optimization of small molecule antagonists of vasoactive intestinal peptide receptor-1 (VIPR1)', BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 22, pagg. 2287-2290.

Srivastava, Neelam ; Mathur, Arvind ; Kayser, Lauren E. ; Karatt, Tajudheen ; K, Kumaragurubaran ; Roy, Amrita ; Cooper, Christopher B. ; Chen, Jing ; Karmakar, Sukhen ; Gupta, Anuradha ; Kong, Yan ; Harikrishnan, Lalgudi S. ; Nirschl, David S. ; Cvijic, Maryellen ; Trainor, George L. ; Poss, Michael A. ; Burford, Neil T. ; Srivastava, Neelam ; Wong, Tai W. / Identification and optimization of small molecule antagonists of vasoactive intestinal peptide receptor-1 (VIPR1). In: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. 2012 ; Vol. 22. pagg. 2287-2290.

@article{b21710dd4ed9435e9ad0af7d938d8ed2,

title = "Identification and optimization of small molecule antagonists of vasoactive intestinal peptide receptor-1 (VIPR1)",

abstract = "Identification, synthesis and structure-activity relationship of small-molecule VIPR1 antagonists encompassing two chemical series are described.",

author = "Neelam Srivastava and Arvind Mathur and Kayser, {Lauren E.} and Tajudheen Karatt and Kumaragurubaran K and Amrita Roy and Cooper, {Christopher B.} and Jing Chen and Sukhen Karmakar and Anuradha Gupta and Yan Kong and Harikrishnan, {Lalgudi S.} and Nirschl, {David S.} and Maryellen Cvijic and Trainor, {George L.} and Poss, {Michael A.} and Burford, {Neil T.} and Neelam Srivastava and Wong, {Tai W.}",

year = "2012",

language = "English",

volume = "22",

pages = "2287--2290",

journal = "BIOORGANIC & MEDICINAL CHEMISTRY LETTERS",

issn = "0960-894X",

}

TY - JOUR

T1 - Identification and optimization of small molecule antagonists of vasoactive intestinal peptide receptor-1 (VIPR1)

AU - Srivastava, Neelam

AU - Mathur, Arvind

AU - Kayser, Lauren E.

AU - Karatt, Tajudheen

AU - K, Kumaragurubaran

AU - Roy, Amrita

AU - Cooper, Christopher B.

AU - Chen, Jing

AU - Karmakar, Sukhen

AU - Gupta, Anuradha

AU - Kong, Yan

AU - Harikrishnan, Lalgudi S.

AU - Nirschl, David S.

AU - Cvijic, Maryellen

AU - Trainor, George L.

AU - Poss, Michael A.

AU - Burford, Neil T.

AU - Srivastava, Neelam

AU - Wong, Tai W.

PY - 2012

Y1 - 2012

N2 - Identification, synthesis and structure-activity relationship of small-molecule VIPR1 antagonists encompassing two chemical series are described.

AB - Identification, synthesis and structure-activity relationship of small-molecule VIPR1 antagonists encompassing two chemical series are described.

UR - http://hdl.handle.net/10447/105375

M3 - Article

VL - 22

SP - 2287

EP - 2290

JO - BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

JF - BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

SN - 0960-894X

ER -

Accesso al documento

OA Link